Chen C, Li X, Neumann CS, Lo MM-C, Schreiber SL. Convergent diversity-oriented synthesis of small-molecule hybrids. Angew Chem Int Ed Engl. 2005;44(15):2249-52. doi:10.1002/anie.200462798.

Strausberg RL, Schreiber SL. From knowing to controlling: a path from genomics to drugs using small molecule probes. Science. 2003;300(5617):294-5. doi:10.1126/science.1083395.

Ong S-E, Li X, Schenone M, Schreiber SL, Carr SA. Identifying cellular targets of small-molecule probes and drugs with biochemical enrichment and SILAC. Methods Mol Biol. 2012;803:129-40. doi:10.1007/978-1-61779-364-6_9.

Koehler AN. A complex task? Direct modulation of transcription factors with small molecules. Curr Opin Chem Biol. 2010;14(3):331-40. doi:10.1016/j.cbpa.2010.03.022.

Corsello SM, Roti G, Ross KN, et al. Identification of AML1-ETO modulators by chemical genomics. Blood. 2009;113(24):6193-205. doi:10.1182/blood-2008-07-166090.

An F. Fluorescence-based assays. Methods Mol Biol. 2009;486:97-107. doi:10.1007/978-1-60327-545-3_7.

Ong S-E, Schenone M, Margolin AA, et al. Identifying the proteins to which small-molecule probes and drugs bind in cells. Proc Natl Acad Sci U S A. 2009;106(12):4617-22. doi:10.1073/pnas.0900191106.

Seiler KP, Kuehn H, Happ MP, Decaprio D, Clemons PA. Using ChemBank to probe chemical biology. Curr Protoc Bioinformatics. 2008;Chapter 14:Unit 14.5. doi:10.1002/0471250953.bi1405s22.

Hyman SE. Revolution stalled. Sci Transl Med. 2012;4(155):155cm11. doi:10.1126/scitranslmed.3003142.

Tibbitt MW, Dahlman JE, Langer R. Emerging Frontiers in Drug Delivery. J Am Chem Soc. 2016;138(3):704-17. doi:10.1021/jacs.5b09974.