Luo T, Schreiber SL. Gold(I)-catalyzed coupling reactions for the synthesis of diverse small molecules using the build/couple/pair strategy. J Am Chem Soc. 2009;131(15):5667-74. doi:10.1021/ja900414s.

Bradner JE, McPherson OM, Koehler AN. A method for the covalent capture and screening of diverse small molecules in a microarray format. Nat Protoc. 2006;1(5):2344-52. doi:10.1038/nprot.2006.282.

Uchida T, Rodriquez M, Schreiber SL. Skeletally diverse small molecules using a build/couple/pair strategy. Org Lett. 2009;11(7):1559-62. doi:10.1021/ol900173t.

Gerard B, O’Shea MW, Donckele E, et al. Application of a catalytic asymmetric Povarov reaction using chiral ureas to the synthesis of a tetrahydroquinoline library. ACS Comb Sci. 2012;14(11):621-30. doi:10.1021/co300098v.

Gray L, Wang X, Brown C, Kuai L, Schreiber SL. Diversity synthesis of complex pyridines yields a probe of a neurotrophic signaling pathway. Org Lett. 2008;10(13):2621-4. doi:10.1021/ol8004936.

Wang Y, Jimenez M, Sheehan P, et al. Selective access to trisubstituted macrocyclic E- and Z-alkenes from the ring-closing metathesis of vinylsiloxanes. Org Lett. 2013;15(6):1218-21. doi:10.1021/ol400134d.

Kim KH, Kim W, Howard TP, et al. SWI/SNF-mutant cancers depend on catalytic and non-catalytic activity of EZH2. Nat Med. 2015;21(12):1491-6. doi:10.1038/nm.3968.

Titov DV, Cracan V, Goodman RP, Peng J, Grabarek Z, Mootha VK. Complementation of mitochondrial electron transport chain by manipulation of the NAD+/NADH ratio. Science. 2016;352(6282):231-5. doi:10.1126/science.aad4017.

Scully SS, Zheng S-L, Wagner BK, Schreiber SL. Synthesis of oxazocenones via gold(I)-catalyzed 8-endo-dig hydroalkoxylation of alkynamides. Org Lett. 2015;17(3):418-21. doi:10.1021/ol503273v.

Chen I, Dorr BM, Liu DR. A general strategy for the evolution of bond-forming enzymes using yeast display. Proc Natl Acad Sci U S A. 2011;108(28):11399-404. doi:10.1073/pnas.1101046108.