An aldol-based build/couple/pair strategy for the synthesis of medium- and large-sized rings: discovery of macrocyclic histone deacetylase inhibitors. Marcaurelle, LA , Comer E. , Dandapani S. , Duvall JR , Gerard B. , Kesavan S. , Lee MD 4th , Liu H. , Lowe JT , Marie JC , Mulrooney CA , Pandya BA , Rowley A. , Ryba TD , Suh BC , Wei J. , Young DW , Akella LB , Ross NT , Zhang YL , et al. Journal of the American Chemical Society, 2010/12/01, Volume 132, Issue 47, p.16962-76, (2010)
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Abstract